Letrozole (Femara) has been touted as one of the three most commonly taken aromatase inhibitors by anabolic steroid users for the effective control of estrogen side effects that are usually caused by the use of amortizing steroids. Besides Letrozole, the two other most commonly used AI’s are non-steroidal Arimidex and steroidal Aromasin. Of these three, the most potent AI’s that can be used against estrogen levels in the body.

What is Letrozole (Femara)?

The main purpose for the development of this drug medication together with all the other AIs, that bodybuilders and athletes use when they take anabolic steroids, has been for the medical treatment of breast cancer in postmenopausal women.

Role of letrozole against estrogen levels

The main reason why this AI is only used in women of this age is because of its powerful ability in blocking the development of estrogen in the body, which would cause serious health issues if used in pre-menopausal women.

For male users of anabolic steroids, the drug’s ability in blocking estrogen development has proved to be very attractive to them, especially in their aim to address the adverse side effects of estrogen when using steroids.

The good news about letrozole is its ability to lower overall estrogen levels by blocking the enzyme aromatase.

Difference between letrozole and SERMs

This is the main difference that letrozole has to all the other popular estrogen control drugs especially for steroid users which are also known as SERMs.

These estrogen control drugs only target very specific areas of the body whereas letrozole focuses on the whole body.

This quality permits Letrozole to work against a wider scope of estrogenic side effects which steroids cause when they are taken. The two main side effects caused by taking steroids is gynecomastia and water retention.

Letrozole also has the ability to prevent the development of high blood pressure that can also accompany excess water retention when left unattended.

Effects of letrozole on Gynecomastia and control of estrogen

The most favorable account of the curing power of letrozole was reported by steroid users who claimed that letrozole has proven so powerful and effective it was able to successfully reverse the effects of gyno when they used the drug.

Still experts hold it would be much better to try and prevent gyno from making a start rather than reversing its progress once it got started. This could have been an unusually lucky break when using letrozole, since normally, once gyno started, it would be irreversible without the use of surgery.

It’s definitely known that this drug medication is capable of reducing the whole circulating levels of estrogen in the body. This is different from what SERM drugs are able to do since they only target specific receptors to bind themselves onto in order to control the progress of gyno.

Letrozole on its part will not only be able to control gyno but would have spare energy to also control water retention, the other main negative effect of taking steroids, which everyone would rather avoid.

During your use of letrozole it’s not unusual to expect your levels of estrogen to be dramatically decreased given that this drug medication is the most powerful AI that you can currently purchase.

As a matter of fact you may find your estrogen level to occasionally drop to very low levels which can prove problematic to the men who require a small amount of estrogen in order to function properly.

It’s very important to remember that during any steroid cycle, the main aim when using an AI is to lower, lessen and finally prevent the side effects of estrogen which will certainly emerge as a result of your taking of steroids that can aromatize.

Other benefits from letrozole control of estrogen

Additional benefits can accrue to you from your use of letrozole such as;

With the strength of letrozole you’d be able to prevent the effects of water retention

Your physique will take on a much more ripped, harder and drier appearance due to the fact that you’re not holding water.

These qualitative outcomes can make letrozole essentially useful as a tool for competitive bodybuilders, whose main goal is to eliminate fluid retention as much as possible and they have the perfect ally in letrozole.

Ideal Letrozole dosages during anabolic steroid use

There’s nothing to be gained from taking too much Letrozole during a steroid cycle when you’re taking steroid. Instead, you’ll only succeed in causing negative side effects such as fatigue. It’s therefore more sensible to maintain a correct dose.

The most commonly used daily dose hovers around 2.5mg per day, so this should be your standard quantitative measurement which you shouldn’t exceed but you can certainly go even lower under it.

It has been found that a low dose range of between 0.5mg to 1.25mg every two days is often sufficient to provide an excellent protection against any estrogenic side effects for most men.

However, if you happen to experience signs of gynecomastia developing, an appropriate step to take would be to increase the dose to about 2.5mg daily may even suffice to reverse the symptoms. Even so, be on the alert for a sudden burst of energy during this change in dosage.

Once you notice that the gyno symptoms have subsided, you should take it as a cue to reduce your letrozole dose back down to the standard estrogenic protection levels.

What of the Letrozole dosage for females?

To be succinctly honest, any increase in estrogen levels, pose no great threat for female steroid users than for male users.

The main reason why females use an AI such as Letrozole would typically be for reducing water retention, especially if they are participating in competitive bodybuilding or athletic performance where a reduction in water retention is highly desirable.

Even so, Letrozole has never been recommended as the first option for females simply because of its potency in greatly minimizing estrogen and therefore not prudent to use in medically treating women who are still in their premenopausal stage.

Nevertheless, women who are determined to take letrozole are cautioned to use a dose of just 0.5mg daily and monitor the results and effects from this dose level.

Bottom line

The post cycle therapy or PCT is the ultimate launching platform from which you can catapult yourself to international fame as a bodybuilder or an athletic performer or forever hold your silence. It is the final stage where the usage of anabolic steroids and AIs and side effects reach their highest peak in athletic endeavor but once successful, bodybuilders and athletics alike will be able to relish the feeling of victory and accomplishment that only the determined and brave can enjoy.